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Co-Regulation of CYP3A4 and CYP3A5 and Contribution to Hepatic and Intestinal Midazolam Metabolism

Molecular Pharmacology · 2002 · Vol. 62(1) · pp. 162–172
Yvonne S. LinAmy L.S. DowlingSean QuigleyFederico M. FarinJiong ZhangJatinder K. LambaErin G. SchuetzKenneth E. Thummel
Pharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsDrug-Induced Hepatotoxicity and ProtectionCYP3A4MidazolamMetabolismDrug metabolismCYP3A5BiologyChemistryPharmacologyCytochrome P450Endocrinology

MeSH terms

AllelesBase SequenceCytochrome P-450 Enzyme SystemGenotypeHumansMixed Function OxygenasesHydroxylationIntestine, SmallMicrosomes, LiverMidazolamMolecular Sequence DataPhenotypeRNA, MessengerSequence Homology, Nucleic AcidAnti-Anxiety Agents
Citations
443
FWCI
30.78
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References
45
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100%
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Co-Regulation of CYP3A4 and CYP3A5 and Contribution to Hepatic and Intestinal Midazolam Metabolism · Scinovex