reviewTop 1% cited
Carbonic anhydrases: novel therapeutic applications for inhibitors and activators
Nature Reviews Drug Discovery · 2008 · Vol. 7(2) · pp. 168–181
Claudiu T. Supuran✉(University of Florence)
Enzyme function and inhibitionCholinesterase and Neurodegenerative DiseasesChemical Reactions and MechanismsLipogenesisPharmacologyDrug discoveryGene isoformChemistryBioinformaticsMedicineBiologyBiochemistryLipid metabolism
MeSH terms
AnimalsCarbonic AnhydrasesCarbonic Anhydrase InhibitorsHumansIsoenzymesModels, MolecularStructure-Activity RelationshipDrug DesignMolecular Structure
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References
Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX
Bioorganic & Medicinal Chemistry Letters · 2003 · 257 citations
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