articleTop 10% cited
Evaluation of Various Dissolution Media for Predicting In Vivo Performance of Class I and II Drugs
Pharmaceutical Research · 1998 · Vol. 15(5) · pp. 698–705
Eric Galia✉Eleftheria Nicolaides(National and Kapodistrian University of Athens)D. Hörter(Goethe University Frankfurt)Raimar Löbenberg(Goethe University Frankfurt)Christos Reppas(National and Kapodistrian University of Athens)Jennifer Dressman(Goethe University Frankfurt)
Drug Solubulity and Delivery SystemsPharmacy and Medical PracticesCrystallization and Solubility StudiesDissolutionChemistryChromatographySolubilityDosage formGastric fluidAqueous mediumAcetaminophenAqueous solutionBiochemistry
MeSH terms
AcetaminophenAnimalsAnti-Inflammatory Agents, Non-SteroidalAntifungal AgentsAntihypertensive AgentsCapsulesDanazolPharmaceutical PreparationsEstrogen AntagonistsKetoconazoleMefenamic AcidMetoprololMilkSolubilityWater
Citations
917
FWCI
8.87
field-weighted impact
References
35
Percentile
99%
vs. same field & year
Citations per year
Cited by
A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System
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Characterization of the Human Upper Gastrointestinal Contents Under Conditions Simulating Bioavailability/Bioequivalence Studies
Pharmaceutical Research · 2005 · 652 citations
Dissolution Media Simulating Conditions in the Proximal Human Gastrointestinal Tract: An Update
Pharmaceutical Research · 2008 · 739 citations
References
Analytical profiles of drug substances
Journal of Pharmaceutical Sciences · 1975 · 1,498 citations
A Theoretical Basis for a Biopharmaceutic Drug Classification: The Correlation of in Vitro Drug Product Dissolution and in Vivo Bioavailability
Pharmaceutical Research · 1995 · 5,270 citations
Upper Gastrointestinal (GI) pH in Young, Healthy Men and Women
Pharmaceutical Research · 1990 · 766 citations
Dissolution Testing as a Prognostic Tool for Oral Drug Absorption: Immediate Release Dosage Forms
Pharmaceutical Research · 1998 · 1,072 citations
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