articleTop 1% cited
Dissolution Media Simulating Conditions in the Proximal Human Gastrointestinal Tract: An Update
Pharmaceutical Research · 2008 · Vol. 25(7) · pp. 1663–1676
Ekarat Jantratid✉(Goethe University Frankfurt)Niels Janssen(Goethe University Frankfurt)Christos Reppas(National and Kapodistrian University of Athens)Jennifer Dressman(Goethe University Frankfurt)
Drug Solubulity and Delivery SystemsGastrointestinal motility and disordersHelicobacter pylori-related gastroenterology studiesPostprandialDissolutionStomachSmall intestineDigestion (alchemy)Gastrointestinal tractChemistryIn vivoHuman stomachBiophysics
MeSH terms
AlgorithmsBileBody FluidsBuffersChemistry, PharmaceuticalChemistry, PhysicalCulture MediaDrug StoragePharmaceutical PreparationsEnzymesExcipientsFastingGastric Acidity DeterminationGastric MucosaHumans
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100%
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References
Evaluation of Various Dissolution Media for Predicting In Vivo Performance of Class I and II Drugs
Pharmaceutical Research · 1998 · 917 citations
Upper Gastrointestinal (GI) pH in Young, Healthy Men and Women
Pharmaceutical Research · 1990 · 766 citations
Dissolution Testing as a Prognostic Tool for Oral Drug Absorption: Immediate Release Dosage Forms
Pharmaceutical Research · 1998 · 1,072 citations
Physicochemical and Physiological Mechanisms for the Effects of Food on Drug Absorption: The Role of Lipids and pH
Journal of Pharmaceutical Sciences · 1997 · 602 citations
Characterization of the Human Upper Gastrointestinal Contents Under Conditions Simulating Bioavailability/Bioequivalence Studies
Pharmaceutical Research · 2005 · 652 citations
THE UNITED STATES PHARMACOPEIA.
Journal of the American Medical Association · 1908 · 1,259 citations
Lipids and lipid-based formulations: optimizing the oral delivery of lipophilic drugs
Nature Reviews Drug Discovery · 2007 · 1,755 citations
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