reviewTop 1% cited
Polymeric Amorphous Solid Dispersions: A Review of Amorphization, Crystallization, Stabilization, Solid-State Characterization, and Aqueous Solubilization of Biopharmaceutical Classification System Class II Drugs
Journal of Pharmaceutical Sciences · 2016 · Vol. 105(9) · pp. 2527–2544
Shrawan Baghel(Waterford Institute of Technology)Helen Cathcart(Waterford Institute of Technology)Niall J. O’Reilly✉(Waterford Institute of Technology)
Drug Solubulity and Delivery SystemsProtein purification and stabilityAnalytical Chemistry and ChromatographyAmorphous solidBiopharmaceuticalSolubilityCrystallizationMaterials scienceCharacterization (materials science)Dispersion (optics)PolymerSupersaturationChemical engineering
MeSH terms
BiopharmaceuticsCrystallizationDrug CarriersDrug StabilityPharmaceutical PreparationsPolymersSolubility
Citations
926
FWCI
49.50
field-weighted impact
References
230
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References
A Theoretical Basis for a Biopharmaceutic Drug Classification: The Correlation of in Vitro Drug Product Dissolution and in Vivo Bioavailability
Pharmaceutical Research · 1995 · 5,270 citations
What is the True Solubility Advantage for Amorphous Pharmaceuticals?
Pharmaceutical Research · 2000 · 1,334 citations
Solid dispersion of poorly water‐soluble drugs: Early promises, subsequent problems, and recent breakthroughs
Journal of Pharmaceutical Sciences · 1999 · 1,638 citations
Supersaturating Drug Delivery Systems: The Answer to Solubility-Limited Oral Bioavailability?
Journal of Pharmaceutical Sciences · 2009 · 915 citations
Manufacturing of solid dispersions of poorly water soluble drugs by spray drying: Formulation and process considerations
International Journal of Pharmaceutics · 2012 · 533 citations
Water Soluble Polymers for Pharmaceutical Applications
Polymers · 2011 · 598 citations
Estimation of Drug–Polymer Miscibility and Solubility in Amorphous Solid Dispersions Using Experimentally Determined Interaction Parameters
Pharmaceutical Research · 2008 · 491 citations
Pharmaceutical Particle Engineering via Spray Drying
Pharmaceutical Research · 2007 · 1,614 citations
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