articleTop 10% cited
Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
Biochemical Pharmacology · 1973 · Vol. 22(23) · pp. 3099–3108
Yung-Chi Cheng✉(Yale University)William H. Prusoff(Yale University)
Receptor Mechanisms and SignalingViral Infectious Diseases and Gene Expression in InsectsProtein purification and stabilityUncompetitive inhibitorNon-competitive inhibitionKineticsEnzyme kineticsSubstrate (aquarium)ChemistryEnzymeStereochemistryActive siteBiochemistry
MeSH terms
Binding, CompetitiveEnzyme InhibitorsKineticsMathematics
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