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Varenicline Is a Partial Agonist at α4β2 and a Full Agonist at α7 Neuronal Nicotinic Receptors

Molecular Pharmacology · 2006 · Vol. 70(3) · pp. 801–805
Nicotinic Acetylcholine Receptors StudyReceptor Mechanisms and SignalingInsect and Pesticide ResearchVareniclinePartial agonistCytisineAgonistPharmacologyNicotinic agonistChemistryReceptorAcetylcholine receptorInternal medicine

MeSH terms

VareniclineAnimalsBenzazepinesNeuronsOocytesQuinoxalinesReceptors, NicotinicXenopus laevisNicotinic AgonistsRatsalpha7 Nicotinic Acetylcholine Receptor

Funding

  • University of Miami
  • U.S. Food and Drug Administration
Citations
552
FWCI
11.00
field-weighted impact
References
26
Percentile
99%
vs. same field & year
Citations per year
References
Varenicline:  An α4β2 Nicotinic Receptor Partial Agonist for Smoking Cessation
Journal of Medicinal Chemistry · 2005 · 930 citations
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