reviewTop 1% cited
How were new medicines discovered?
Nature Reviews Drug Discovery · 2011 · Vol. 10(7) · pp. 507–519
David C. Swinney✉(Roche (United States))Jason Anthony(Roche (United States))
Computational Drug Discovery MethodsBiotechnology and Related FieldsBioinformatics and Genomic NetworksDrug discoveryFood and drug administrationDrugPhenotypic screeningMedicinePharmacologyComputational biologyMechanism (biology)Small moleculeDrug development
MeSH terms
Pharmacological PhenomenaDrug IndustryDrug Evaluation, PreclinicalHumansUnited StatesUnited States Food and Drug AdministrationDrug DesignDrug ApprovalDrug DiscoveryMolecular Targeted TherapyDrug-Related Side Effects and Adverse Reactions
Citations
1,768
FWCI
140.64
field-weighted impact
References
175
Percentile
100%
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References
Enzyme Structure and Mechanism
FEBS Letters · 1978 · 760 citations
Discovery and development of bevacizumab, an anti-VEGF antibody for treating cancer
Nature Reviews Drug Discovery · 2004 · 2,577 citations
How many drug targets are there?
Nature Reviews Drug Discovery · 2006 · 3,473 citations
Aripiprazole, a Novel Antipsychotic, Is a High-Affinity Partial Agonist at Human Dopamine D2 Receptors
Journal of Pharmacology and Experimental Therapeutics · 2002 · 915 citations
Varenicline: An α4β2 Nicotinic Receptor Partial Agonist for Smoking Cessation
Journal of Medicinal Chemistry · 2005 · 930 citations
Maraviroc (UK-427,857), a Potent, Orally Bioavailable, and Selective Small-Molecule Inhibitor of Chemokine Receptor CCR5 with Broad-Spectrum Anti-Human Immunodeficiency Virus Type 1 Activity
Antimicrobial Agents and Chemotherapy · 2005 · 1,144 citations
Heparin and Low-Molecular-Weight Heparin Mechanisms of Action, Pharmacokinetics, Dosing, Monitoring, Efficacy, and Safety
CHEST Journal · 2001 · 1,571 citations
Cell Signaling by Receptor Tyrosine Kinases
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