article Open AccessTop 10% cited
Potent and selective inhibitors of the proteasome: Dipeptidyl boronic acids
Bioorganic & Medicinal Chemistry Letters · 1998 · Vol. 8(4) · pp. 333–338
Julian Adams✉Mark L. Behnke(Allscripts (United States))Shaowu Chen(Allscripts (United States))Amy Cruickshank(Allscripts (United States))Lawrence R. Dick(Allscripts (United States))Louis Grenier(Allscripts (United States))Janice M. Klunder(Allscripts (United States))Yu-Ting Ma(Allscripts (United States))Louis Plamondon(Allscripts (United States))Ross L. Stein(Allscripts (United States))
Ubiquitin and proteasome pathwaysPeptidase Inhibition and AnalysisProtein Degradation and InhibitorsChemistryBoronic acidProteasomePotencyCombinatorial chemistryAldehydeBiochemistryPharmacologyStereochemistryIn vitro
MeSH terms
Boronic AcidsCysteine EndopeptidasesMultienzyme ComplexesProtease InhibitorsMolecular StructureProteasome Endopeptidase Complex
Citations
680
FWCI
5.28
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References
20
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96%
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References
Lange's handbook of chemistry
Choice Reviews Online · 1992 · 7,155 citations
STRUCTURE AND FUNCTIONS OF THE 20S AND 26S PROTEASOMES
Annual Review of Biochemistry · 1996 · 2,423 citations
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