reviewTop 1% cited
Sulfoximines from a Medicinal Chemist's Perspective: Physicochemical and in vitro Parameters Relevant for Drug Discovery
European Journal of Medicinal Chemistry · 2016 · Vol. 126 · pp. 225–245
Marcus Frings(RWTH Aachen University)Carsten Bolm(RWTH Aachen University)Andreas Blum(Boehringer Ingelheim (Germany))Christian Gnamm✉(Boehringer Ingelheim (Germany))
Synthesis and Catalytic ReactionsPharmacogenetics and Drug MetabolismEpigenetics and DNA MethylationChemistryDrug discoveryMoietySolubilityCombinatorial chemistryMetabolic stabilitySulfonamideStereochemistryComputational biologyOrganic chemistry
MeSH terms
Chemistry, PharmaceuticalHumansSulfur CompoundsChemical PhenomenaDrug Discovery
Citations
470
FWCI
29.56
field-weighted impact
References
96
Percentile
100%
vs. same field & year
Citations per year
References
New N- and O-arylations with phenylboronic acids and cupric acetate
Tetrahedron Letters · 1998 · 1,138 citations
Copper-Promoted Carbon-Heteroatom Bond Cross-Coupling with Boronic Acids and Derivatives
Synthesis · 2010 · 550 citations
New aryl/heteroaryl CN bond cross-coupling reactions via arylboronic acid/cupric acetate arylation
Tetrahedron Letters · 1998 · 1,043 citations
Sulfoximines: Structures, Properties and Synthetic Applications
Synthesis · 2000 · 397 citations
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