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SR 144528, the First Potent and Selective Antagonist of the CB2 Cannabinoid Receptor

Journal of Pharmacology and Experimental Therapeutics · 1998 · Vol. 284(2) · pp. 644–650

M Rinaldi-Carmona✉(Sanofi (France))Francis Barth(Sanofi (France))J Millan(Sanofi (France))Jean‐Marie Derocq(Sanofi (France))Pierre Casellas(Sanofi (France))Christian Congy(Sanofi (France))Didier Oustric(Sanofi (France))M Sarran(Sanofi (France))Monsif Bouaboula(Sanofi (France))Bernard Calandra(Sanofi (France))M Portier(Sanofi (France))David Shire(Sanofi (France))J. C. BrelièreGérard Le Fur(Sanofi (France))

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Cannabis and Cannabinoid Research Neurotransmitter Receptor Influence on Behavior Diet, Metabolism, and DiseaseCannabinoid receptor type 2ReceptorCannabinoid receptorCannabinoidAdenylyl cyclaseAgonistChemistryGPR18PharmacologyAntagonist

MeSH terms

Cyclic AMPAdenylyl CyclasesAdministration, OralAnimalsB-LymphocytesCamphanesCannabinoidsCyclohexanolsCricetinaeHumansLymphocyte ActivationPyrazolesReceptors, DrugRecombinant ProteinsCHO Cells

Citations

704

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37.34

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100%

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References

Refinement of the Coomassie blue method of protein quantitation

Analytical Biochemistry · 1978 · 1,585 citations

Determination and characterization of a cannabinoid receptor in rat brain.

Molecular Pharmacology · 1988 · 2,412 citations

Comparison of the pharmacology and signal transduction of the human cannabinoid CB1 and CB2 receptors.

Molecular Pharmacology · 1995 · 877 citations

Expression of Central and Peripheral Cannabinoid Receptors in Human Immune Tissues and Leukocyte Subpopulations

European Journal of Biochemistry · 1995 · 1,747 citations

Transformation of rat cells by DNA of human adenovirus 5

Virology · 1973 · 660 citations

SR141716A, a potent and selective antagonist of the brain cannabinoid receptor

FEBS Letters · 1994 · 1,747 citations

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