articleTop 10% cited
Allosteric Modulation of the Cannabinoid CB1 Receptor
Molecular Pharmacology · 2005 · Vol. 68(5) · pp. 1484–1495
M. R. Price✉(University of Aberdeen)Gemma L. Baillie(University of Aberdeen)Adèle Thomas(University of Aberdeen)Lesley StevensonMorag Easson(Merck (Japan))Richard Goodwin(Merck (Japan))Adèle McLean(Merck (Japan))Lorraine McIntosh(Merck (Japan))Gillian Goodwin(Merck (Japan))Glenn Walker(Merck (Japan))Paul Westwood(Merck (Japan))Julia Marrs(Merck (Japan))Fiona Thomson(Merck (Japan))Phillip M. Cowley(Merck (Japan))Arthur Christopoulos(University of Melbourne)Roger G. Pertwee(University of Aberdeen)Ruth A. Ross(University of Aberdeen)
Cannabis and Cannabinoid ResearchNeuroscience and Neuropharmacology ResearchNeurotransmitter Receptor Influence on BehaviorAllosteric regulationRadioligandInverse agonistChemistryAllosteric modulatorStereochemistryAgonistAmideReceptorCooperativity
MeSH terms
RimonabantAllosteric RegulationAnimalsBinding SitesCyclohexanolsHumansMalePiperidinesPyrazolesVas DeferensGuanosine 5'-O-(3-Thiotriphosphate)Receptor, Cannabinoid, CB1Mice
Citations
443
FWCI
10.77
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References
39
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99%
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References
Anandamide and vanilloid TRPV1 receptors
British Journal of Pharmacology · 2003 · 595 citations
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