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Discovery of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV-1 agents

Bioorganic & Medicinal Chemistry Letters · 2001 · Vol. 11(13) · pp. 1793–1796
Maria Letizia BarrecaAlba ChimirriLaura De LucaAnna‐Maria MonfortePietro MonforteAngela RaoMaria ZappalàJan BalzariniErik De ClercqChristophe PannecouqueMyriam Witvrouw
HIV/AIDS drug development and treatmentHIV Research and TreatmentHepatitis C virus researchChemistryIn vitroHuman immunodeficiency virus (HIV)StereochemistryChemical synthesisNucleosideNucleotidyltransferaseStructure–activity relationshipCombinatorial chemistryBiochemistry

MeSH terms

Structure-Activity RelationshipThiazolesVirus ReplicationHIV-1Reverse Transcriptase InhibitorsAnti-HIV Agents
Citations
236
FWCI
2.62
field-weighted impact
References
10
Percentile
89%
vs. same field & year
Citations per year
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