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[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain.
Journal of Pharmacology and Experimental Therapeutics · 1989 · Vol. 251(3) · pp. 888–893
Michael F. Jarvis✉(Novartis (Switzerland))Richard SchulzA. HutchisonU HMatthew A. SillsMichael Williams
Adenosine and Purinergic SignalingPharmacological Receptor Mechanisms and EffectsSynthesis and Characterization of Heterocyclic CompoundsCGS-21680AdenosineAdenosine receptorAgonistAdenosine A2A receptorCCPAChemistryBinding siteReceptorStereochemistry
MeSH terms
AdenosineAnimalsBinding, CompetitiveBrainCorpus StriatumPhenethylaminesRadioligand AssayReceptors, PurinergicTritiumAdenosine-5'-(N-ethylcarboxamide)RatsIn Vitro Techniques
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546
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